5 Results for "

AG221

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "AG221" in MCE Product Catalog:

17
17 Cited Publications
Cat. No.: HY-18690
CAS No.: 1446502-11-9
Synonyms: AG-221
Research Areas:  

Cancer

Enasidenib is an oral, potent, reversible, selective inhibitor of the IDH2 mutant enzymes, with IC50s of 100 and 400 nM against IDH2 R140Q and IDH2 R172K, respectively.
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17
17 Cited Publications
Cat. No.: HY-18690A
CAS No.: 1650550-25-6
Synonyms: AG-221 mesylate
Research Areas:  

Cancer

Enasidenib mesylate is a first-in-class, oral, potent, reversible, selective inhibitor of the IDH2 mutant enzymes.
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Cat. No.: HY-18690R
CAS No.: 1446502-11-9
Synonyms: AG-221 (Standard)
Enasidenib (Standard) is the analytical standard of Enasidenib. This product is intended for research and analytical applications. Enasidenib is an oral, potent, reversible, selective inhibitor of the IDH2 mutant enzymes, with IC50s of 100 and 400 nM against IDH2R140Q and IDH2R172K, respectively.
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Cat. No.: HY-18690AR
CAS No.: 1650550-25-6
Synonyms: AG-221 mesylate (Standard)
Enasidenib (mesylate) (Standard) is the analytical standard of Enasidenib (mesylate). This product is intended for research and analytical applications. Enasidenib mesylate is a first-in-class, oral, potent, reversible, selective inhibitor of the IDH2 mutant enzymes.
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Cat. No.: HY-18690S
CAS No.: 2095569-76-7
Synonyms: AG-221-d6
Enasidenib-d6 (AG-221-d6) is the deuterium labeled Enasidenib (HY-18690) . Enasidenib is an oral, potent, reversible, selective inhibitor of the IDH2 mutant enzymes, with IC50s of 100 and 400 nM against IDH2 R140Q and IDH2 R172K, respectively .
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