1 Result for "

APL5125

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "APL5125" in MCE Product Catalog:

Cat. No.: HY-178980
CAS No.: 2830619-57-1
Target:  

Casein Kinase

Research Areas:  

Cancer

APL-5125 (Compound 61f) is a potent, selective and orally active ATP-competitive CK2α inhibitor with an IC50 of 0.348 nM and a Ki of 0.095 nM. APL-5125 binds to CK2α in a bivalent manner, simultaneously interacting with the ATP-binding site and the αD pocket. APL-5125 exhibits antitumor activity and can be used for the research of cancer, such as colon cancer .
loading...
    loading...