1 Result for "

BMS-986180

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "BMS-986180" in MCE Product Catalog:

Cat. No.: HY-150080
CAS No.: 1803444-21-4
Synonyms: BMS-986180
Target:  

HIV HIV Integrase

Research Areas:  

Infection

GSK3739936 (BMS-986180) is a potent HIV-1 allosteric integrase inhibitor with an IC50 value of 11.1 nM and an EC50 value of 1.7 nM. GSK3739936 is also a weak CYP inhibitor (IC50>24.3 μM). GSK3739936 shows favorable pharmacokinetic property in preclinical species with rapid absorption, low to moderate clearance and excellent oral bioavailability .
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