2 Results for "

BMS204352

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "BMS204352" in MCE Product Catalog:

Cat. No.: HY-108584
CAS No.: 187523-35-9
Purity:  99.56%
Synonyms: BMS-204352
Target:  

Potassium Channel

Research Areas:  

Neurological Disease

Flindokalner (BMS-204352) is a potassium channel modulator. Flindokalner is a positive modulator of all neuronal Kv7 channel subtypes expressed in HEK293 cells. Flindokalner is also a large conductance calcium-activated K channel (BKca) positive modulator. Flindokalner shows a negative modulatory activity at Kv7.1 channels (Ki=3.7 μM), and acts as a negative modulator of GABAA receptors. Flindokalner shows anxiolytic efficacy in vivo .
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Cat. No.: HY-108584R
CAS No.: 187523-35-9
Synonyms: BMS-204352 (Standard)
Flindokalner (Standard) is the analytical standard of Flindokalner. This product is intended for research and analytical applications. Flindokalner (BMS-204352) is a potassium channel modulator. Flindokalner is a positive modulator of all neuronal Kv7 channel subtypes expressed in HEK293 cells. Flindokalner is also a large conductance calcium-activated K channel (BKca) positive modulator. Flindokalner shows a negative modulatory activity at Kv7.1 channels (Ki=3.7 μM), and acts as a negative modulator of GABAA receptors. Flindokalner shows anxiolytic efficacy in vivo .
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