1 Result for "

DETQ

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "DETQ" in MCE Product Catalog:

Cat. No.: HY-115553
CAS No.: 1638667-81-8
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

DETQ is a selective, allosteric and orally active dopamine D1 receptor (Dopamine Receptor) potentiator. In HEK293 cells expressing the human D1 receptor, DETQ increases cAMP with an EC50 of 5.8 nM and a Kb of 26 nM. DETQ shows ~30-fold less potent at rat and mouse D1 receptors and is inactive at the human D5 receptor .
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