1 Result for "

FK3657

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "FK3657" in MCE Product Catalog:

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Cat. No.: HY-15791
CAS No.: 167838-64-4
Synonyms: FK-3657
Target:  

Bradykinin Receptor

Research Areas:  

Inflammation/Immunology

FR173657 is an orally active bradykinin B2 receptor antagonist (IC50: 0.56, 1.5, 2.9 nM for pig, rat, human B2 receptor respectively). FR173657 (p.o.) inhibits BK-induced bronchoconstriction in guinea-pigs (ED50: 0.075 mg/kg). FR173657 (p.o.) also inhibits Carrageenin-induced paw oedema in mice (ED50: 6.8 mg/kg). FR173657 can be used for research of inflammatory disease .
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