1 Result for "

GPA512

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "GPA512" in MCE Product Catalog:

Cat. No.: HY-123827
CAS No.: 1808115-35-6
Target:  

STAT Drug Intermediate

Research Areas:  

Cancer

GPA512 is an orally active STAT3 inhibitor and a prodrug of Galiellalactone (HY-125170). GPA512 inhibits the binding of STAT3 to DNA, downregulates STAT3-activated genes, and suppresses tumor growth in prostate cancer xenograft models. GPA512 is rapidly converted to Galiellalactone in plasma. GPA512 can be used in research related to castration-resistant prostate cancer .
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