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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
6 Results for "
HM30181
" in MedChemExpress (MCE) Product Catalog:
Products (6)
6 Results for "HM30181" in MCE Product Catalog:
5
5 Cited Publications
Synonyms: HM30181; HM30181A
Target:
Research Areas:
Encequidar (HM30181; HM30181A) is a potent and selective inhibitor of P-glycoprotein.
5
5 Cited Publications
Synonyms: HM30181 mesylate; HM30181A mesylate
Target:
Research Areas:
Encequidar mesylate (HM30181 mesylate; HM30181A mesylate) is a competitive and potent P-glycoprotein inhibitor.
Cat. No.: HY-13646R
CAS No.: 849675-66-7
Synonyms: HM30181 (Standard); HM30181A (Standard)
Target:
Research Areas:
Encequidar (Standard) is the analytical standard of Encequidar. This product is intended for research and analytical applications. Encequidar (HM30181; HM30181A) is a potent and selective inhibitor of P-glycoprotein.
Cat. No.: HY-13646C
CAS No.: 2097125-58-9
Synonyms: HM30181 mesylate hydrochloride; HM30181A mesylate hydrochloride
Target:
Research Areas:
Encequidar (HM30181) mesylate hydrochloride is a potent and selective inhibitor of P-glycoprotein (MDR1). Encequidar mesylate hydrochloride improves anti-tumor efficacy of Paclitaxel (HY-B0015) in mouse tumor models .
Cat. No.: HY-13646B
CAS No.: 849675-88-3
Synonyms: HM30181 hydrochloride; HM30181A hydrochloride
Target:
Research Areas:
Encequidar hydrochloride (HM30181 hydrochloride) is an oral P-glycoprotein (P-gp) inhibitor with the activity of enhancing the oral bioavailability of P-gp substrate drugs. Encequidar shows the highest potency among various MDR1 inhibitors, with IC50=0.63nM. Encequidar effectively blocks the transepithelial transport of paclitaxel in MDCK monolayer cells, with IC50=35.4nM .
Cat. No.: HY-13646AR
CAS No.: 849675-87-2
Synonyms: HM30181 mesylate (Standard); HM30181A mesylate (Standard)
Target:
Research Areas:
Encequidar (mesylate) (Standard) is the analytical standard of Encequidar (mesylate). This product is intended for research and analytical applications. Encequidar mesylate (HM30181 mesylate; HM30181A mesylate) is a competitive and potent P-glycoprotein inhibitor.
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Protocols
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