1 Result for "

M2-adrenoceptor

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "M2-adrenoceptor" in MCE Product Catalog:

Cat. No.: HY-106874B
CAS No.: 119813-87-5
Synonyms: rel-RS-15385-197
Target:  

Adrenergic Receptor

Research Areas:  

Neurological Disease

rel-Delequamine (rel-RS-15385-197) is an orally active, brain-penetrant, potent and selective M2-adrenoceptor antagonist and α2-adrenoceptor antagonist. rel-Delequamine has a pKi of 9.45 for α2-adrenoceptors in the rat cortex. rel-Delequamine augments K +-evoked release of noradrenaline with an EC50 of 1 nM .
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