1 Result for "

M4 mAChR Modulator-1

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "M4 mAChR Modulator-1" in MCE Product Catalog:

  • Targets Recommended:
Cat. No.: HY-159177
Target:  

mAChR

Research Areas:  

Neurological Disease

M4 mAChR Modulator-1 (compound 23i) is a M4 mAChR positive allosteric modulator (PAM). M4 mAChR Modulator-1 exhibits significantly greater cooperativity with ACh in β-arrestin recruitment over G protein activation. M4 mAChR Modulator-1 displays weak PAM effect in G protein-mediated responses, but strong PAM effect in β-arrestin recruitment .
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