M4 mAChR Modulator-1
M4 mAChR Modulator-1 (compound 23i) is a M4 mAChR positive allosteric modulator (PAM). M4 mAChR Modulator-1 exhibits significantly greater cooperativity with ACh in β-arrestin recruitment over G protein activation. M4 mAChR Modulator-1 displays weak PAM effect in G protein-mediated responses, but strong PAM effect in β-arrestin recruitment.
For research use only. We do not sell to patients.
- Formula: C22H23N5O
- Molecular Weight:373.45
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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mAChR4 |
Chemical Information
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Molecular Weight 373.45
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Formula C22H23N5O
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SMILES
O=C1NCC2=C1C=C(C3=NC(C)=NC=C3C4=CN(CC5CCCC5)N=C4)C=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
M4 mAChR Modulator-1 Related Classifications
HY-159177 Related Classifications
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