1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. mAChR
  4. mAChR5 Isoform

mAChR5

 

mAChR5 Related Products (4):

Cat. No. Product Name Effect Purity
  • HY-107651
    VU 0365114
    Agonist 99.51%
    VU 0365114 is a selective mAChR M5 positive allosteric modulator, with an EC50 of 2.7 μM, and >30 μM for M1, M2, M3 and M4 receptors.
  • HY-148502
    VU6019650
    Antagonist
    VU6019650 is a potent and selective orthosteric antagonist of M5 mAChR (IC50=36 nM), can be used for opioid use disorder (OUD) relief.
  • HY-107656
    PTAC oxalate
    Modulator
    PTAC oxalate is a selective muscarinic receptor ligand.
  • HY-148527
    LAS190792
    Antagonist
    LAS190792 (AZD8999) is a potent muscarinic antagonist and β2-adrenoceptor agonist with pIC50 8.9, 8.8, 8.8, 9.2, 8.2, 7.5, 9.1, 5.6 for M1, M2, M3, M4, M5, β1, β2, β3, respectively.