2. Signaling Pathways
  3. GPCR/G Protein
    Neuronal Signaling
  4. mAChR
  5. mAChR3 Isoform

mAChR3

 

mAChR3 Related Products (13):

Cat. No. Product Name Effect Purity
  • HY-76772
    Cevimeline hydrochloride hemihydrate
    		Agonist ≥98.0%
    Cevimeline hydrochloride hemihydrate (SNI-2011) is a quinuclidine derivative of acetylcholine and a selective and orally active muscarinic M1 and M3 receptor agonist.
  • HY-12980
    Batefenterol
    		Antagonist 98.30%
    Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively.
  • HY-107647
    (S)-(+)-Dimethindene maleate
    		Antagonist 99.94%
    (S)-(+)-Dimethindene maleate, an enantiomer, is a potent M2-selective muscarinic receptor antagonist (pA2 = 7.86/7.74; pKi = 7.78).
  • HY-32067
    Aceclidine
    		Modulator ≥98.0%
    Aceclidine is a modulator of M3 muscarinic acetylcholine receptor.
  • HY-14825A
    Tarafenacin D-tartrate
    		Antagonist 99.87%
    Tarafenacin D-tartrate (SVT-40776 D-tartrate) is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over M2 receptor.
  • HY-P4156
    VLVNTFCDSCIPKTYWNLGY TFA
    VLVNTFCDSCIPKTYWNLGY TFA is an antigenic peptide of M3 muscarinic receptor (M3R).
  • HY-101679A
    YM-58790 free base
    		Antagonist
    YM-58790 free base is a potent antagonist of mAChR.
  • HY-107656
    PTAC oxalate
    		Modulator
    PTAC oxalate is a selective muscarinic receptor ligand.
  • HY-B1332
    Ipratropium bromide hydrate
    		Antagonist 98.50%
    Ipratropium bromide (Sch 1000) hydrate is a muscarinic receptor antagonist, with IC50s of 2.9 nM, 2 nM, and 1.7 nM for M1, M2, and M3 receptors, respectively.
  • HY-100958
    4-DAMP
    		Antagonist 99.87%
    4-DAMP is a potent antagonist of M3 receptor and also has a high affinity for the closely-related M5 receptor.
  • HY-14825
    Tarafenacin
    		Antagonist
    Tarafenacin(SVT-40776) is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over M2 receptor.
  • HY-101679
    YM-58790
    		Antagonist
    YM-58790 is a potent antagonist of mAChR.
  • HY-148527
    LAS190792
    		Antagonist
    LAS190792 (AZD8999) is a potent muscarinic antagonist and β2-adrenoceptor agonist with pIC50 8.9, 8.8, 8.8, 9.2, 8.2, 7.5, 9.1, 5.6 for M1, M2, M3, M4, M5, β1, β2, β3, respectively.