1. GPCR/G Protein
    Neuronal Signaling
  2. Dopamine Receptor
    Serotonin Transporter
  3. Deschloroclozapine

Deschloroclozapine 

Cat. No.: HY-42110 Purity: 99.79%
Handling Instructions

Deschloroclozapine is a dual dopamine and serotonin receptor antagonist with Kis of 200, 2500, 420, 39, 84, 40 nM for dopamine D1, D2,D4, and serotonin S2A, S2C, S3, respectively.

For research use only. We do not sell to patients.

Deschloroclozapine Chemical Structure

Deschloroclozapine Chemical Structure

CAS No. : 1977-07-7

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Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 110 In-stock
Estimated Time of Arrival: December 31
10 mg USD 100 In-stock
Estimated Time of Arrival: December 31
50 mg USD 350 In-stock
Estimated Time of Arrival: December 31
100 mg USD 550 In-stock
Estimated Time of Arrival: December 31
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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

Deschloroclozapine is a dual dopamine and serotonin receptor antagonist with Kis of 200, 2500, 420, 39, 84, 40 nM for dopamine D1, D2,D4, and serotonin S2A, S2C, S3, respectively.

IC50 & Target

Ki: 200 nM (Dopamne D1), 2500 nM (Dopamne D2), 420 nM (Dopamne D4), 39 nM (Serotonin S2A), 84 nM (Serotonin S2C), 200 nM (Serotonin S3)[1]

Molecular Weight

292.38

Formula

C₁₈H₂₀N₄

CAS No.

1977-07-7

SMILES

CN1CCN(C2=NC3=CC=CC=C3NC4=CC=CC=C42)CC1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : ≥ 83.3 mg/mL (284.90 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 3.4202 mL 17.1010 mL 34.2021 mL
5 mM 0.6840 mL 3.4202 mL 6.8404 mL
10 mM 0.3420 mL 1.7101 mL 3.4202 mL
*Please refer to the solubility information to select the appropriate solvent.
References
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Keywords:

DeschloroclozapineDopamine ReceptorSerotonin Transporter5-HTTSERTSLC6A4Inhibitorinhibitorinhibit

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Deschloroclozapine
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HY-42110
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