1 Result for "

MK5596

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "MK5596" in MCE Product Catalog:

Cat. No.: HY-10575
CAS No.: 1044586-68-6
Research Areas:  

Metabolic Disease

MK-5596 is an efficient, selective and orally active CB1R (IC50 = 1.0 nM, EC50 = 5.8 nM) inverse agonist. MK-5596 has weak hERG inhibitory activity. MK-5596 has strong weight loss and appetite suppression effects. MK-5596 has a certain inhibitory effect on CYP enzymes (CYP3A4: IC50 = 3.3 μM, CYP2C8: IC50 = 11 μM, CYP2C9: IC50 = 18 μM, CYP2D6: IC50 = 6 μM). MK-5596 can be used for research on conditions such as obesity .
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