1 Result for "

OP1690

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "OP1690" in MCE Product Catalog:

Cat. No.: HY-181345
Target:  

Estrogen Receptor/ERR

Research Areas:  

Cancer

OP-1690 is a complete estrogen receptor (ERα) antagonist (CERAN), with pIC50 values of 7.5 and 7.9 in alkaline phosphatase (AP) activity assay and TR-FRET assay, respectively. OP-1690 modulates receptor function by inducing ERα tetramerization, effectively induces ERα degradation, inhibits target gene transcription, but exhibits low antiproliferative potency. OP-1690 can be used for breast cancer research .
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