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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
3 Results for "
PROTAC CBP/P300 Degrader-4
" in MedChemExpress (MCE) Product Catalog:
Products (3)
3 Results for "PROTAC CBP/P300 Degrader-4" in MCE Product Catalog:
Cat. No.: HY-183802
Target:
Research Areas:
PROTAC CBP/P300 Degrader-4 is a p300/CBP PROTAC degrader with DC50 of 17.4 nM and 10.2 nM against p300 and CBP in U2OS cells, respectively. PROTAC CBP/P300 Degrader-4 forms ternary complexes with p300 or CBP and an E3 ligase, drives ubiquitination, and mediates proteasomal degradation. PROTAC CBP/P300 Degrader-4 can be used for the research of hematological malignancies .
Cat. No.: HY-183817
CAS No.: 2484742-13-2
Research Areas:
GNE-781-COOH is a CBP/p300 degrader. GNE-781-COOH also acts as a ligand for target protein for PROTAC (Ligands for Target Protein for PROTAC), which can be used to synthesize PROTAC CBP/P300 Degrader-4 (HY-183802) .
Cat. No.: HY-183818
Target:
Research Areas:
CRBN ligand-903 is a CRBN-binding ligand as well as a ligand for E3 ubiquitin ligase (Ligands for E3 Ligase). CRBN ligand-903 can be used to synthesize PROTAC CBP/P300 Degrader-4 (HY-183802) .
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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
