1 Result for "

SR-0813

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "SR-0813" in MCE Product Catalog:

Cat. No.: HY-145409
CAS No.: 2597186-19-9
Purity:  99.93%
Research Areas:  

Cancer

SR-0813 is a potent and selective ENL/AF9 YEATS domain inhibitor. SR-0813 has IC50 and EC50 values of 25 nM and 205 nM for ENL YEATS domain, respectively. SR-0813 has IC50 and EC50 values of 311 nM and 76 nM (CETSA) for AF9 YEATS domain, respectively. SR-0813 binds MAP3K19 with over 100-fold lower affinity (Kd=3.5 μM) than ENL YEATS (Kd=30 nM). SR-0813 can be used for the research of acute leukemia .
loading...
    loading...