1 Result for "

TA0201

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "TA0201" in MCE Product Catalog:

Cat. No.: HY-124234
CAS No.: 169679-53-2
Target:  

Endothelin Receptor

Research Areas:  

Cardiovascular Disease

TA-0201 is a novel orally active, competitive, non-peptide endothelin receptor antagonist. TA-0201 antagonizes the specific binding of [ 125I]ET-1 to cloned human receptors of ETA and ETB with Ki values of 15 pM and 41 nM, respectively. TA-0201 inhibits the pressor response to the exogenous big ET-1 .
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