1 Result for "

TRK851

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "TRK851" in MCE Product Catalog:

Cat. No.: HY-16979
CAS No.: 189015-24-5
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

RK-851 is a highly selective and orally active δ-opioid receptor antagonist, with a negative logarithm of the antagonist concentration (pA2) of 8.84. TRK-851 exhibits the selectivity for the δ receptor of more than 100 times higher than that for the μ or κ receptors. TRK-851 exhibits a potent antitussive effect in a rat model of capsaicin-induced cough. TRK-851 can be used for research on antitussive effects .
loading...
    loading...