1 Result for "

TRKAF589L

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "TRKAF589L" in MCE Product Catalog:

  • Isoforms Recommended:
Cat. No.: HY-149965
CAS No.: 2924344-29-4
Target:  

Trk Receptor Apoptosis

Research Areas:  

Cancer

TRK-IN-23 (compound 24b) is a potent and orally active TRK inhibitor with IC50 values of 0.5 nM, 9 nM, 14 nM, 4.4 nM, and 4.8 nM against TRKA, TRKC, TRKA G595R, TRKA F589L, and TRKA G667C, respectively. TRK-IN-23 indues apoptosis of Ba/F3-TRKAG595Rand Ba/F3-TRKAG667C cells .
loading...
    loading...