1 Result for "

Tipepidine citrate

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "Tipepidine citrate" in MCE Product Catalog:

Cat. No.: HY-B2185
CAS No.: 14698-07-8
Tipepidine citrate is a non-narcotic antitussive agent. Tipepidine citrate reversibly inhibits dopamine D2 receptor-mediated GIRK current (IDA(GIRK)), thereby activating VTA dopamine neurons, with an IC50 of 7.0 μM for IDA(GIRK). Tipepidine activates AMPK. Tipepidine citrate has antidepressant-like effects. Tipepidine citrate enhances the analgesic effect of Carbamazepine (HY-B0246). Tipepidine citrate improves adipose tissue fibrosis and glucose intolerance in high-fat diet-induced obese mice .
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