2 Results for "

U62066

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "U62066" in MCE Product Catalog:

Cat. No.: HY-106756
CAS No.: 87151-85-7
Synonyms: U-62066
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Spiradoline (U-62066), an arylacetamide, is a selective kappa opioid receptor (KOR) agonist with a Ki of 8.6 nM in guinea pig. The Ki values of Spiradoline for μ and δ receptors are 252 nM and 9400 nM, respectively. Spiradoline has potent diuretic, analgesic, antiarrythmic, antitussive, neuroprotective properties and easily penetrates the blood-brain barrier .
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Cat. No.: HY-124959
CAS No.: 87173-97-5
Purity:  99.81%
Synonyms: U-62066 mesylate
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Spiradoline mesylate (U-62066 mesylate), an arylacetamide, is a selective kappa opioid receptor (KOR) agonist with a Ki of 8.6 nM in guinea pig. The Ki values of Spiradoline mesylate for μ and δ receptors are 252 nM and 9400 nM, respectively. Spiradoline mesylate has potent diuretic, analgesic, antiarrythmic, antitussive, neuroprotective properties and easily penetrates the blood-brain barrier .
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