1 Result for "

cellular class IIa HDAC activity

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "cellular class IIa HDAC activity" in MCE Product Catalog:

Cat. No.: HY-184524
CAS No.: 3035189-46-6
Target:  

PROTACs HDAC

Research Areas:  

Others

PROTAC HDAC4 Degrader-2 is a class IIa selective negative control for HDAC4 PROTAC degraders, with an IC50 of 0.15 μM against HDAC4 and a cellular IC50 of 0.18 μM. PROTAC HDAC4 Degrader-2 fails to effectively recruit the VHL E3 ligase, and thus does not induce significant degradation of HDAC4 protein .
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