1 Result for "

tetrapeptide aldehyde

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "tetrapeptide aldehyde" in MCE Product Catalog:

Cat. No.: HY-P10007
CAS No.: 159659-05-9
Synonyms: Z-GPFL-CHO
Target:  

Proteasome

Research Areas:  

Cancer

Z-Gly-Pro-Phe-Leu-CHO (Z-GPFL-CHO) is a tetrapeptide aldehyde that acts as a highly selective and potent proteasomal inhibitor (Ki = 1.5 µM for branched chain amino acid preferring, 2.3 µM for small neutral amino acid preferring, and 40.5 µM for chymotrypsin-like activities; IC50 = 3.1 µM for peptidyl-glutamyl peptide hydrolyzing activity) .
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