34099-70-2
Chemical Structure
M1 receptor modulator-1
- CAS No.: 34099-70-2
- Formula:C15H11BrN2S
- Molecular Weight:331.23
InChIKey: RGEBXTAQYWVMJZ-UHFFFAOYSA-N
SMILES: S=C1NC2=C(C(C3=CC=CC=C3)=NC1)C=C(Br)C=C2
Biological Activity: M1 receptor modulator-1 is a low-efficacy positive allosteric modulator of the muscarinic M1 receptor (mAChR1), with an EC50 of 71 nM for the human M1 receptor. M1 receptor modulator-1 enables use-dependent attenuation of neurotransmitter signals and exhibits excellent in vivo properties without pseudo-agonist activity. M1 receptor modulator-1 can be used in research related to Alzheimer's disease and schizophrenia[1].
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M1 receptor modulator-1 | M1 receptor modulator-1 is a low-efficacy positive allosteric modulator of the muscarinic M1 receptor (mAChR1), with an EC50 of 71 nM for the human M1 receptor. M1 receptor modulator-1 enables use-dependent attenuation of neurotransmitter signals and exhibits excellent in vivo properties without pseudo-agonist activity. M1 receptor modulator-1 can be used in research related to Alzheimer's disease and schizophrenia. | |||||||||||||||||||||
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Keywords
