1176326-78-5
1176326-78-5
Chemical Structure
DSP-1053 benzenesulfonate
- CAS No.: 1176326-78-5
- Formula:C32H38BrNO7S
- Molecular Weight:660.62
IUPAC Name: 6-(2-(4-(4-bromo-3-(2-methoxyethoxy)benzyl)piperidin-1-yl)ethyl)chroman-4-one benzenesulfonate
InChIKey: UVZRSKPRJFFXHO-UHFFFAOYSA-N
SMILES: O=C1CCOC2=CC=C(CCN3CCC(CC4=CC=C(Br)C(OCCOC)=C4)CC3)C=C12.O=S(C5=CC=CC=C5)(O)=O
Biological Activity: DSP-1053, a benzylpiperidine derivative, is a potent serotonin transporter (SERT) inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity[1].
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DSP-1053 benzenesulfonate | DSP-1053, a benzylpiperidine derivative, is a potent serotonin transporter (SERT) inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity. | |||||||||||||||||||||
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References
Keywords
