DSP-1053 benzenesulfonate
DSP-1053, a benzylpiperidine derivative, is a potent serotonin transporter (SERT) inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity.
For research use only. We do not sell to patients.
- CAS No.: 1176326-78-5
- Formula: C32H38BrNO7S
- Molecular Weight:660.62
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT1A Receptor |
5-HT1A Receptor 5.05 nM (Ki) |
Chemical Information
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CAS No. 1176326-78-5
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Molecular Weight 660.62
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Formula C32H38BrNO7S
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SMILES
O=C1CCOC2=CC=C(CCN3CCC(CC4=CC=C(Br)C(OCCOC)=C4)CC3)C=C12.O=S(C5=CC=CC=C5)(O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)