2134675-36-6
Chemical Structure
Ziftomenib
Synonym(s): KO-539
- CAS No.: 2134675-36-6
- Formula:C33H42F3N9O2S2
- Molecular Weight:717.87
IUPAC Name: (S)-4-methyl-5-((4-((2-(methylamino)-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl)amino)piperidin-1-yl)methyl)-1-(2-(4-(methylsulfonyl)piperazin-1-yl)propyl)-1H-indole-2-carbonitrile
InChIKey: BGGALFIXXQOTPY-NRFANRHFSA-N
SMILES: N#CC(N1C[C@@H](N2CCN(S(=O)(C)=O)CC2)C)=CC3=C1C=CC(CN4CCC(NC5=C(C=C(CC(F)(F)F)S6)C6=NC(NC)=N5)CC4)=C3C
Biological Activity: Ziftomenib (KO-539) is an orally active menin-MLL interaction inhibitor with antitumor activities (WO2017161028A1, compound 151)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Ziftomenib | 99.43% | Ziftomenib (KO-539) is an orally active menin-MLL interaction inhibitor with antitumor activities (WO2017161028A1, compound 151). | ||||||||||||||||||||
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Ziftomenib (Standard) | ≥98% | Ziftomenib (Standard) is the analytical standard of Ziftomenib (HY-132001). This product is intended for research and analytical applications. Ziftomenib (KO-539) is an orally active menin-MLL interaction inhibitor with antitumor activities (WO2017161028A1, compound 151). | ||||||||||||||||||||
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Ziftomenib-d4 | Ziftomenib-d4 (KO-539-d4) is the deuterium labeled Ziftomenib (HY-132001). Ziftomenib (KO-539) is an orally active menin-MLL interaction inhibitor with antitumor activities. | |||||||||||||||||||||
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Ziftomenib-d3 | Ziftomenib-d3 (KO-539-d3) is the deuterium labeled Ziftomenib (HY-132001). Ziftomenib (KO-539) is an orally active menin-MLL interaction inhibitor with antitumor activities. | |||||||||||||||||||||
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-
Similarity Score 1.00
HY-132001A(R)-Ziftomenib -
Similarity Score 0.76
HY-136360MI-3454 -
Similarity Score 0.67
HY-117365MI-1481 -
Similarity Score 0.65
HY-16925MI-503 -
Similarity Score 0.61
HY-160018BAY-155 -
Similarity Score 0.59
HY-19809MI-463 -
Similarity Score 0.57
HY-19810MI-538 -
Similarity Score 0.53
HY-19319MI-136 -
Similarity Score 0.53
HY-172416Balomenib -
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