620112-78-9
620112-78-9
Chemical Structure
CCG-63802
- CAS No.: 620112-78-9
- Formula:C26H18N4O2S
- Molecular Weight:450.51
IUPAC Name: (E)-2-(benzo[d]thiazol-2-yl)-3-(9-methyl-4-oxo-2-(m-tolyloxy)-4H-pyrido[1,2-a]pyrimidin-3-yl)acrylonitrile
InChIKey: VFSVKVQMZDJFQX-NBVRZTHBSA-N
SMILES: N#C/C(C1=NC2=CC=CC=C2S1)=C\C3=C(N=C4C(C)=CC=CN4C3=O)OC5=CC=CC(C)=C5
Biological Activity: CCG-63802 is a selective, reversible and allosteric RGS4 inhibitor. CCG-63802 specifically binds to RGS4 and blocks the RGS4-Gαo interaction, with an IC50 value of 1.9 μM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CCG-63802 | 98.83% | CCG-63802 is a selective, reversible and allosteric RGS4 inhibitor. CCG-63802 specifically binds to RGS4 and blocks the RGS4-Gαo interaction, with an IC50 value of 1.9 μM. | ||||||||||||||||||||
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References
Keywords
