2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. GABA Receptor
  4. CGP44532

CGP44532 is a GABAB receptor agonist with a pEC50 (geometric mean of the half-maximal effective concentration) value of 5.63 μM.

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CGP44532

CGP44532 構造式

CAS 番号 : 133345-68-3

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CGP44532 関連抗体

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製品説明

CGP44532 is a GABAB receptor agonist with a pEC50 (geometric mean of the half-maximal effective concentration) value of 5.63 μM[1].

Cellular Effect
Cell Line Type Value Description References
CHO-K1 EC50
600 nM
Compound: (R)-4
Agonist activity at human recombinant GABABreceptor expressed in CHO-K1 cells assessed as inhibition of intracellular calcium release by FLIPR
Agonist activity at human recombinant GABABreceptor expressed in CHO-K1 cells assessed as inhibition of intracellular calcium release by FLIPR
[PMID: 18578471]
Oocyte IC50
5.4 μM
Compound: R(+)-CGP-44533
Antagonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp method
Antagonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp method
[PMID: 17981464]
分子量

153.12

分子式

C4H12NO3P
CAS 番号
SMILES

O=P(C)(C[C@H](O)CN)O
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
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CGP44532 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CGP44532133345-68-3CGP 44532CGP-44532GABA ReceptorGamma-aminobutyric acid Receptorγ-Aminobutyric acid Receptorantiepilepticcognitive-enhancementanalgesicantidepressantInhibitorinhibitorinhibit

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製品名:
CGP44532
製品番号:
HY-116197
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