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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
87 Results for "
Benzamides
" in MedChemExpress (MCE) Product Catalog:
Products (87)
87 Results for "Benzamides" in MCE Product Catalog:
11
11 Publications Verification
Art. -Nr.: HY-B1019
CAS. Nr.: 15676-16-1
Target:
Forschungsgebiete:
Sulpiride is an orally active dopamine D2/D3 receptor antagonist. Sulpiride is an atypical antipsychotic agent of the benzamide family. Sulpiride can be used in research into anxiety, depression and breast cancer .
9
9 Cited Publications
Target:
Forschungsgebiete:
Raclopride is a dopamine D2/D3 receptor antagonist with potential antipsychotic effects. Raclopride binds to D2 and D3 receptors with Kis of 1.8 nM and 3.5 nM, respectively .
5
5 Cited Publications
Forschungsgebiete:
CX546 is a first-generation and selective benzamide-type positive AMPAR modulator. CX546 is a prototypical ampakine agent and has antipsychotic effects .
2
Target:
Forschungsgebiete:
Azasetron (Y-25130) hydrochloride, a benzamide derivative, is a potent and selective 5-HT3 receptor antagonist. Azasetron is used in the study for Chemotherapy-induced nausea and vomiting (CINV) .
1
Target:
Forschungsgebiete:
Levosulpiride (RV-12309) is the (S)-enantiomer of sulpiride, which is a D2 receptor a antagonist, an atypical antipsychotic agent of the benzamide class.
1
1 Cited Publications
Synonyms: Benzenecarboxamide; Phenylamide
Category:
Alkaloids Human Gut Microbiota Metabolites Other Alkaloids Other Diseases Endogenous metabolite Disease Research Fields
Target:
Art. -Nr.: HY-P4070
CAS. Nr.: 1188379-43-2
Target:
Forschungsgebiete:
Art. -Nr.: HY-145819
CAS. Nr.: 2669785-85-5
JPS036 is a benzamide-based Von Hippel-Lindau (VHL) E3-ligase proteolysis targeting chimeras (PROTAC). JPS036 degrades class I histone deacetylase (HDAC). JPS036 is potent HDAC1/2 degrader correlated with greater total differentially expressed genes and enhanced apoptosis in HCT116 cells .
Art. -Nr.: HY-147342
CAS. Nr.: 156724-91-3
Target:
Forschungsgebiete:
β-Benzamide adenine dinucleotide is a biologically active metabolite of benzamide riboside. β-Benzamide adenine dinucleotide is a competitive inhibitor of human NAD kinase with a Ki value of 90 μM, and inhibits human IMPDH with IC50 values of 0.787 μM and 0.884 μM for type I and type II, respectively. β-Benzamide adenine dinucleotide exhibits inhibitory activities against lactate dehydrogenase, glutamate dehydrogenase, and malate dehydrogenase. β-Benzamide adenine dinucleotide can be used for the study of chronic myelogenous leukemia .
Art. -Nr.: HY-112547
CAS. Nr.: 1034297-58-9
Synonyms: CRT0066051
CRT5, a pyrazine benzamide, is a potent and selective inhibitor for all three isoforms of PKD in endothelial cells treated with VEGF (IC50s = 1, 2, and 1.5 nM for PKD1, PKD2, and PKD3, respectively). CRT5 decreases VEGF-induced endothelial migration, proliferation and tubulogenesis .
Art. -Nr.: HY-B1019R
CAS. Nr.: 15676-16-1
Target:
Forschungsgebiete:
Sulpiride (Standard) is the analytical standard of Sulpiride. This product is intended for research and analytical applications. Sulpiride is an orally active dopamine D2/D3 receptor antagonist. Sulpiride is an atypical antipsychotic agent of the benzamide family. Sulpiride can be used in research into anxiety, depression and breast cancer .
Art. -Nr.: HY-145815A
Reinheit: 98.40%
JPS014 TFA is a benzamide-based Von Hippel-Lindau (VHL) E3-ligase proteolysis targeting chimeras (PROTAC). JPS014 TFA degrades class I histone deacetylase (HDAC). JPS014 TFA is potent HDAC1/2 degrader correlated with greater total differentially expressed genes and enhanced apoptosis in HCT116 cells .
Art. -Nr.: HY-W000887
CAS. Nr.: 180516-87-4
Art. -Nr.: HY-Z0283S
CAS. Nr.: 31656-62-9
Synonyms: Benzenecarboxamide-15N; Phenylamide-15N
Art. -Nr.: HY-108976
CAS. Nr.: 98185-20-7
Target:
Forschungsgebiete:
Raclopride tartrate is a selective dopamine D2/D3 receptor antagonist with potential antipsychotic effects. Raclopride tartrate binds to D2 and D3 receptors with Kis of 1.8 nM and 3.5 nM, respectively .
Synonyms: (-)-Remoxipride hydrochloride
Target:
Forschungsgebiete:
(S)-Remoxipride ((-)-Remoxipride) hydrochloride is a selective dopamine D2-receptor antagonist with an IC50 value of 1.57 μM. (S)-Remoxipride hydrochloride can be used for the research of psychotic disorder .
Art. -Nr.: HY-75637
CAS. Nr.: 31230-17-8
Target:
Forschungsgebiete:
2-Amino-N-(pyridin-3-ylmethyl)benzamide is a drug intermediate for synthesis of various active compounds.
Art. -Nr.: HY-W055845
CAS. Nr.: 19227-13-5
Target:
Forschungsgebiete:
4-Methylbenzamide oxime is a model of benzamide oxime and can be used as a substrate for mitochondrial amidoxime reducing component (mARC) catalytic enzyme reduction .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
