Azapetine
Azapetine is an α-adrenergic receptor antagonist, with a IC50 of 0.205 μM against rat α1-adrenergic receptors and a IC50 of 1.3 μM against rat α2-adrenergic receptors. Azapetine blocks α1/α2-adrenergic receptor-mediated contraction of blood vessels and vascular smooth muscles. Azapetine can be used for the research of peripheral vascular diseases.
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- CAS No.: 146-36-1
- Formule: C17H17N
- Masse moléculaire:235.32
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Activité biologique
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rat α1-adrenergic receptor 0.205 μM (IC50) |
rat α2-adrenergic receptor 1.3 μM (IC50) |
Azapetine (45-60 min) exhibits higher binding affinity for α1-adrenergic receptors than for α2-adrenergic receptors in isolated rat brain cell membranes, with an IC50 of 0.205 μM for α1-adrenergic receptors and 1.3 μM for α2-adrenergic receptors[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 146-36-1
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Masse moléculaire 235.32
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Formule C17H17N
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SMILES
C=CCN1CC2=C(C3=C(C1)C=CC=C3)C=CC=C2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Azapetine Related Classifications
HY-181635 Related Classifications
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