146-36-1
146-36-1
Chemical Structure
Azapetine
- CAS No.: 146-36-1
- Formula:C17H17N
- Molecular Weight:235.32
InChIKey: NYGHGTMKALXFIA-UHFFFAOYSA-N
SMILES: C=CCN1CC2=C(C3=C(C1)C=CC=C3)C=CC=C2
Biological Activity: Azapetine is an α-adrenergic receptor antagonist, with a IC50 of 0.205 μM against rat α1-adrenergic receptors and a IC50 of 1.3 μM against rat α2-adrenergic receptors. Azapetine blocks α1/α2-adrenergic receptor-mediated contraction of blood vessels and vascular smooth muscles. Azapetine can be used for the research of peripheral vascular diseases[1].
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Azapetine | Azapetine is an α-adrenergic receptor antagonist, with a IC50 of 0.205 μM against rat α1-adrenergic receptors and a IC50 of 1.3 μM against rat α2-adrenergic receptors. Azapetine blocks α1/α2-adrenergic receptor-mediated contraction of blood vessels and vascular smooth muscles. Azapetine can be used for the research of peripheral vascular diseases. | |||||||||||||||||||||
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References
Keywords
