LG-120907
LG-120907 is a selective androgen receptor (AR) antagonist with a Ki value of 26 nM. LG-120907 inhibits Testosterone-induced increases in ventral prostate (VP) tissue weight and seminal vesicles (SV) tissue weight in vivo.
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- CAS No.: 201654-12-8
- 화학식: C15H13F3N2O
- 분자량:294.28
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- 순도&문서
- References
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Help & FAQs
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CV-1 | IC50 |
27 nM
Compound: 1
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Antagonist activity at human androgen receptor expressed in CV1 cells
Antagonist activity at human androgen receptor expressed in CV1 cells
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[PMID: 17257838] |
| CV-1 | IC50 |
390 nM
Compound: 36
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Antagonistic activity against human progesterone receptor B (hPR-B) in co-transfected CV-1 cells.
Antagonistic activity against human progesterone receptor B (hPR-B) in co-transfected CV-1 cells.
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[PMID: 9484511] |
| CV-1 | IC50 |
58 nM
Compound: 36
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Antagonistic activity against human androgen receptor (hAR) in co-transfected CV-1 cells.
Antagonistic activity against human androgen receptor (hAR) in co-transfected CV-1 cells.
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[PMID: 9484511] |
Chemical Information
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CAS No. 201654-12-8
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분자량 294.28
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화학식 C15H13F3N2O
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SMILES
O=C1C=C(C2=CC=3C=CC(NC3C=C2N1)(C)C)C(F)(F)F
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LG-120907 Related Classifications
HY-119436 Related Classifications
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