2 Results for "

53772-82-0

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "53772-82-0" in MCE Product Catalog:

Cat. No.: HY-184837
CAS No.: 53772-82-0
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

cis-Flupenthixol is an orally active dopamine receptor antagonist, with a Ki value of 1.4 nM for the Dopamine D-1 receptor and 0.74 nM for the Dopamine D-2 receptor. cis-Flupenthixol blocks dopamine receptors in the medial preoptic area and striatum, impairs male mating behavior, and reduces the concentrations of striatal dopamine metabolites. cis-Flupenthixol alters striatal acetylcholine concentrations in a time-dependent manner and enhances Apomorphine (HY-12723)-induced stereotyped behaviors. cis-Flupenthixol inhibits exploratory locomotor activity and triggers a compensatory increase in dopamine turnover in the striatum and limbic regions. cis-Flupenthixol can be used in studies related to tardive dyskinesia .
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Cat. No.: HY-W654197
CAS No.: 1246833-30-6
(E/Z)-Flupentixol dihydrochloride-d4 is the deuterium labeled (E/Z)-Flupentixol dihydrochloride.
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