1246833-30-6
1246833-30-6
Chemical Structure
(E/Z)-Flupentixol dihydrochloride-d4
- CAS No.: 1246833-30-6
- Formula:C23H21D4F3N2OS
- Molecular Weight:438.54
IUPAC Name: (Z)-2-(4-(3-(2-(trifluoromethyl)-9H-thioxanthen-9-ylidene)propyl)piperazin-1-yl)ethan-1,1,2,2-d4-1-ol
InChIKey: NJMYODHXAKYRHW-VASCPITCSA-N
SMILES: OC([2H])(C([2H])(N1CCN(CC/C=C2C3=C(SC4=C\2C=CC=C4)C=CC(C(F)(F)F)=C3)CC1)[2H])[2H]
Biological Activity: (E/Z)-Flupentixol dihydrochloride-d4 is the deuterium labeled (E/Z)-Flupentixol dihydrochloride.
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(E/Z)-Flupentixol dihydrochloride-d4 | (E/Z)-Flupentixol dihydrochloride-d4 is the deuterium labeled (E/Z)-Flupentixol dihydrochloride. | |||||||||||||||||||||
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cis-Flupenthixol | cis-Flupenthixol is an orally active dopamine receptor antagonist, with a Ki value of 1.4 nM for the Dopamine D-1 receptor and 0.74 nM for the Dopamine D-2 receptor. cis-Flupenthixol blocks dopamine receptors in the medial preoptic area and striatum, impairs male mating behavior, and reduces the concentrations of striatal dopamine metabolites. cis-Flupenthixol alters striatal acetylcholine concentrations in a time-dependent manner and enhances Apomorphine (HY-12723)-induced stereotyped behaviors. cis-Flupenthixol inhibits exploratory locomotor activity and triggers a compensatory increase in dopamine turnover in the striatum and limbic regions. cis-Flupenthixol can be used in studies related to tardive dyskinesia. | |||||||||||||||||||||
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