2 Results for "

A71915

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "A71915" in MCE Product Catalog:

Cat. No.: HY-P2026
CAS No.: 132956-87-7
A 71915 is a highly potent and competitive natriuretic peptide receptor A (ANP, NPRA) antagonist (pKi= 9.18). A 71915 displaces [ 125I]ANP dose dependently, with a Ki of 0.65 nM. A71915( pA2= 9.48) against rat ANP-induced cGMP production in NB-OK-1 cells .
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Cat. No.: HY-P1980
Target:  

Apoptosis

Research Areas:  

Metabolic Disease

A-71915 (TFA) is a selective inhibitor of ANP receptor (atrial natriuretic peptide-receptor), induces apoptosis and decreases insulin secretion in RINm5F pancreatic β-cells .
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