1 Result for "

CH5164840

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "CH5164840" in MCE Product Catalog:

Cat. No.: HY-15990
CAS No.: 1052645-73-4
Target:  

HSP

Research Areas:  

Cancer

CH5164840 (16) shows high binding affinity for N-terminal Hsp90a (Kd = 0.52 nM) and strong anti-proliferative activity against human cancer cell lines (HCT116 IC50 = 0.15 μM, NCI-N87 IC50 = 0.066 μM). CH5164840 (16) is orally active (t1/2 = 2.64 h) with potent antitumor efficacy .
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