1 Result for "

CNS-selective

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "CNS-selective" in MCE Product Catalog:

Cat. No.: HY-136207
CAS No.: 2454492-41-0
Purity:  98.4%
Target:  

nAChR

Research Areas:  

Neurological Disease

TC-2559 idifumarate is a CNS-selective, orally active α4β2 subtype of nicotinic acetylcholine receptor (nAChR) partial agonist (EC50=0.18 μM). TC-2559 difumarate shows selectivity for α4β2 over α2β4, α4β4 and α3β4 receptors, with EC50s in the range of 10-30 µM. Antinociceptive effect .
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