1 Result for "

EN1441

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "EN1441" in MCE Product Catalog:

Cat. No.: HY-173626
CAS No.: 2196448-47-0
Target:  

Androgen Receptor

Research Areas:  

Cancer

EN1441 is a covalent degrader targeting the androgen receptor (AR) with an EC50 value of 4.2 μM and its truncated variant AR-V7. EN1441 selectively and potently degrades both AR and AR-V7 in androgen-independent prostate cancer cells. EN1441 is promising for research of androgen-independent prostate cancers .
loading...
    loading...