1 Result for "

EXQ-2d

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "EXQ-2d" in MCE Product Catalog:

Cat. No.: HY-168925
Target:  

Wnt PARP β-catenin

Research Areas:  

Cancer

EXQ-2d is the inhibitor for tankyrase and inhibits TNKS1 and TNKS2 with an IC50 of 48.8 nM and 13.8 nM (pIC50=7.31 and 7.86). EXQ-2d inhibits WNT/β-catenin signaling pathway with IC50 of 515 nM. EXQ-2d exhibits anti-proliferative activity in cancer cells COLO 320DM and RKO with GI50 of 4.9 μM and 77 μM .
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