3 Results for "

GW4064

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "GW4064" in MCE Product Catalog:

57
57 Cited Publications
Cat. No.: HY-50108
CAS No.: 278779-30-9
Target:  

FXR Autophagy

Research Areas:  

Metabolic Disease Cancer

GW 4064 is a potent FXR agonist with an EC50 of 65 nM.
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Cat. No.: HY-50108A
CAS No.: 1089660-72-9
Target:  

FXR

Research Areas:  

Others

(E)-GW 4064 is a FXR agonist .
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Cat. No.: HY-175516
Target:  

FXR PPAR

Research Areas:  

Inflammation/Immunology

dual FXR/PPARδ agonist-2 is a FXR/PPARδ dual agonist through hybridation of FXR agonist GW-4064 and PPARδ agonist GW-0742.dual FXR/PPARδ agonist-2 displays potent dual-target activities with a FXR agonistic EC50 of 12.28 nM and 69 % PPARδ activation at 100 nM. dual FXR/PPARδ agonist-2 shows anti-fibrotic effects in pulmonary fibrosis mouse model .
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