2 Results for "

Indantadol

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Indantadol" in MCE Product Catalog:

Cat. No.: HY-101440A
CAS No.: 202914-18-9
Synonyms: CHF-3381
Target:  

iGluR Monoamine Oxidase

Research Areas:  

Neurological Disease

Indantadol hydrochloride (CHF-3381) is an orally active, non-selective NMDA antagonist and MAO inhibitor. Indantadol hydrochloride blocks the binding of [³H]-MK-801 to NMDA receptors in a non-competitive manner, with an IC50 of 8.1 μM. Indantadol hydrochloride completely inhibits dopamine release caused by NMDA. Indantadol hydrochloride protects neurons, with an ED₅₀ of 35 μM. Indantadol hydrochloride has anticonvulsant and anti-high pain hypersensitivity activities .
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Cat. No.: HY-101440
CAS No.: 202844-10-8
Synonyms: CHF-3381 free base
Target:  

iGluR Monoamine Oxidase

Research Areas:  

Neurological Disease

Indantadol (the free base of CHF-3381) is an orally active, non-selective NMDA antagonist and MAO inhibitor. Indantadol blocks the binding of [³H]-MK-801 to NMDA receptors in a non-competitive manner, with an IC50 of 8.1 μM. Indantadol completely inhibits dopamine release caused by NMDA. Indantadol protects neurons, with an ED₅₀ of 35 μM. Indantadol has anticonvulsant and anti-high pain hypersensitivity activities .
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