2 Results for "

Lei-Dab7

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Lei-Dab7" in MCE Product Catalog:

Cat. No.: HY-P1424
CAS No.: 1061556-49-7
Target:  

Potassium Channel

Research Areas:  

Neurological Disease

Lei-Dab7 is a potent and selective SK2 (KCa2.2) channels blocker with a Kd of 3.8 nM. Lei-Dab7 shows low or no activity on KCa1, KCa3, Kv and Kir2.1 channels .
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Cat. No.: HY-P1424A
Target:  

Potassium Channel

Research Areas:  

Neurological Disease

Lei-Dab7 TFA is a high affinity, selective KCa2.2 (SK2) channel blocker (Kd=3.8 nM). Lei-Dab7 TFA exhibits >200-fold selectivity for KCa2.2 over KCa2.1, KCa2.3, KCa3.1, Kv and Kir2.1. Lei-Dab7 TFA increases theta-burst responses and increases LTP in rat hippocampal slices in vitro.
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