3 Results for "

Masupirdine

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Masupirdine" in MCE Product Catalog:

Cat. No.: HY-109118A
CAS No.: 1791396-46-7
Purity:  99.62%
Synonyms: SUVN-502 mesylate
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally active, and brain-penetrating 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine mesylate has pro-cognitive effects on all stages of cognition (acquisition, consolidation, and retention), and can reverse Scopolamine (HY-N0296), MK-801 (HY-15084B)-induced and aging-related memory deficits. Masupirdine mesylate can be used in the research of Alzheimer's disease .
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Cat. No.: HY-109118
CAS No.: 701205-60-9
Synonyms: SUVN-502 free base
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Masupirdine free base (SUVN-502 free base) is a potent, selective, orally active, and brain-penetrating 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine free base has pro-cognitive effects on all stages of cognition (acquisition, consolidation, and retention), and can reverse Scopolamine (HY-N0296), MK-801 (HY-15084B)-induced and aging-related memory deficits. Masupirdine free base can be used in the research of Alzheimer's disease .
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Cat. No.: HY-109118AR
CAS No.: 1791396-46-7
Synonyms: SUVN-502 mesylate (Standard)
Research Areas:  

Neurological Disease

Masupirdine mesylate (Standard) is the analytical standard of Masupirdine (mesylate) (HY-109118A). This product is intended for research and analytical applications. Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally active, and brain-penetrating 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine mesylate has pro-cognitive effects on all stages of cognition (acquisition, consolidation, and retention), and can reverse Scopolamine (HY-N0296), MK-801 (HY-15084B)-induced and aging-related memory deficits. Masupirdine mesylate can be used in the research of Alzheimer's disease .
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