1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor
  3. Masupirdine free base

Masupirdine free base (Synonyms: SUVN-502 free base)

Cat. No.: HY-109118
Handling Instructions

Masupirdine free base (SUVN-502 free base) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine free base (SUVN-502 free base) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease.

For research use only. We do not sell to patients.

Masupirdine free base Chemical Structure

Masupirdine free base Chemical Structure

CAS No. : 701205-60-9

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Description

Masupirdine free base (SUVN-502 free base) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine free base (SUVN-502 free base) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease[1].

IC50 & Target

Ki: 2.04 nM (human 5-HT6 receptor)[1]

Molecular Weight

478.40

Formula

C₂₁H₂₄BrN₃O₃S

CAS No.

701205-60-9

SMILES

O=S(N1C2=CC=C(OC)C=C2C(CN3CCN(C)CC3)=C1)(C(C=CC=C4)=C4Br)=O

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Masupirdine free base
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HY-109118
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