1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor
  3. Masupirdine mesylate

Masupirdine mesylate (Synonyms: SUVN-502 mesylate)

Cat. No.: HY-109118A
Handling Instructions

Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine mesylate (SUVN-502 mesylate) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease.

For research use only. We do not sell to patients.

Masupirdine mesylate Chemical Structure

Masupirdine mesylate Chemical Structure

CAS No. : 1791396-46-7

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 1107 In-stock
Estimated Time of Arrival: December 31
1 mg USD 150 In-stock
Estimated Time of Arrival: December 31
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10 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine mesylate (SUVN-502 mesylate) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease[1].

IC50 & Target

5-HT6 Receptor

2.04 nM (Ki)

Molecular Weight

670.61

Formula

C₂₃H₃₂BrN₃O₉S₃

CAS No.

1791396-46-7

SMILES

CS(=O)(O)=O.O=S(N1C2=CC=C(OC)C=C2C(CN3CCN(C)CC3)=C1)(C(C=CC=C4)=C4Br)=O.CS(=O)(O)=O

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
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Masupirdine mesylate
Cat. No.:
HY-109118A
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