2 Results for "

Sec61α subunit

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Sec61α subunit" in MCE Product Catalog:

Cat. No.: HY-P87069
Synonyms: chunp6898 antibody; fb62c11 antibody; HSec61 antibody; protein transport protein Sec61 alpha subunit antibody; protein transport protein Sec61 subunit alpha antibody; Protein transport protein Sec61 subunit alpha isoform 1 antibody; S61A1_HUMAN antibody; Sec 61 antibody; Sec 61A antibody; Sec61 alpha 1 antibody; chunp6898 antibody; fb62c11 antibody; HSec61 antibody; protein transport protein Sec61 alpha subunit antibody; protein transport protein Sec61 subunit alpha antibody; Protein transport protein Sec61 subunit alpha isoform 1 antibody; S61A1_HUMAN antibody; Sec 61 antibody; Sec 61A antibody; Sec61 alpha 1 antibody; Sec61 alpha 1 subunit antibody; Sec61 alpha 1 subunit (S. cerevisiae) antibody; Sec61 alpha-1 antibody; Sec61 antibody; Sec61 homolog antibody; Sec61A1 antibody; Sec61aa antibody;

Host:  

Rabbit

Application:  

WB, IHC-P

Reactivity:  

Human, Mouse, Rat

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Cat. No.: HY-P10466
CAS No.: 2377734-91-1
KZR-8445, a cyclic depsipeptide, is a client-selective Sec61 inhibitor. KZR-8445 binds to the fully opened Sec61 lateral gate, blocks lumenal plug domain access, stabilizes lateral gate helices, traps select signal peptides, and disrupts secretory and membrane protein biogenesis. KZR-8445 inhibits pro-inflammatory cytokine secretion in primary immune cells. KZR-8445 inhibits SARS-CoV-2 replication, virus-induced cytotoxicity, and spike protein biogenesis. KZR-8445 blocks disease progression in a mouse model of rheumatoid arthritis. KZR-8445 can be used for the researches of rheumatoid arthritis and SARS-CoV-2 infection .
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