2 Results for "

VB-Caco-2

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "VB-Caco-2" in MCE Product Catalog:

Cat. No.: HY-168742
Target:  

Vasopressin Receptor

Research Areas:  

Neurological Disease

V1a/V2 antagonist 1 (Compound 18j) is an orally active dual V1a and V2 receptor antagonist with high binding affinity for both receptors (Ki: 0.13 nM for hV1a, 0.53 nM for hV2 and 0.5 nM for mV1a; IC50: 2.2 nM for hV1a). V1a/V2 antagonist 1 inhibits Oxytocin (HY-17571)-induced scratching behavior in mice .
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Cat. No.: HY-181551
CAS No.: 2027497-52-3
Target:  

MCHR1 (GPR24)

Research Areas:  

Metabolic Disease

RGH-706 is an orally active, blood-brain barrier-permeable, selective MCH1 receptor antagonist with an IC50 of 6.2 nM against hMCHR1. RGH-706 shows no antagonistic activity against hMCH2 receptors. RGH-706 improves obesity. RGH-706 can be used in research related to obesity and Prader-Willi syndrome .
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